|
C Le Manach, A T Nchinda, T Paquet, D Gonzalez Cabrera, Y Y Adam, Z Han, S Bashyam, M Zabiulla, D Taylor, N Lawrence, K L White, S A Charman, D Waterson, M J Witty, S Wittlin, M E Botha, S H Nondaba, J Reader, L - M Birkholtz, M B Jimenez-Diaz, M S Martínez-Martínez, S Ferrer-Bazaga, I Angulo-Barturen, S Meister, Y Antonova-Koch, E A Winzeler, L J Street, K Chibale (2016) Identification of a potential anti-malarial drug candidate from a series of 2-aminopyrazines by optimization of aqueous solubility and potency across the parasite life-cycle. J. Med. Chem. 59: 21. 9890-9905 Nov 10. |
B Baragaña, N R Norcross, C Wilson, A Porzelle, I Hallyburton, R Grimaldi, M Osuna-Cabello, S Norval, J Riley, L Stojanovski, F R C Simeons, P G Wyatt, M J Delves, S Meister, S Duffy, V M Avery, E A Winzeler, R E Sinden, S Wittlin, J A Frearson, D W Gray, A H Fairlamb, D Waterson, S F Campbell, P Willis, K D Read, I H Gilbert (2016) Discovery of a quinoline-4-carboxamide derivative with a novel mechanism of action, multi-stage antimalarial activity, and potent in vivo efficacy. Journal of Medicinal Chemistry 59: 21. 9672-9685 Sept 10. |
 Alice E Williamson, Paul M Ylioja, Murray N Robertson, Yevgeniya Antonova-Koch, Vicky Avery, Jonathan Baell, Harikrishna Batchu, Sanjay Batra, Jeremy N Burrows, Soumya Bhattacharyya, Felix Calderon, Susan A e Charman, Julie Clark, Benigno Crespo, Matin Dean, Stefan L Debbert, Michael Delves, Adelaide S M Dennis, Frederik Deroose, Sandra Duffy, Sabine Fletcher, Guri Giaever, Irene Hallyburton, Francisco-Javier Gamo, Marinella Gebbia, R Kiplin Guy, Zoe Hungerford, Kiaran Kirk, Maria J Lafuente-Monasterio, Anna Lee, Stephan Meister, Corey Nislow, John P Overington, George Papadatos, Luc Patiny, James Pham, Stuart Ralph, Andrea Ruecker, Eileen Ryan, Christopher Southan, Kumkum Srivastava, Chris Swain, Matthew J Tarnowski, Patrick Thomson, Peter Turner, Iain M Wallace, Timothy N C Wells, Karen White, Laura White, Paul Willis, Elizabeth A Winzeler, Sergio Wittlin, Matthew H Todd (2016) Open Source Drug Discovery - Highly Potent Antimalarial Compounds Derived from the Tres Cantos Arylpyrroles ACS Cent. Sci. 2: 10. 687-701 Sept 26. |
 Wesley C Van Voorhis, John H Adams, Roberto Adelfio, Vida Ahyong, Myles H Akabas, Pietro Alano, Aintzane Alday, Yesmalie Alemán Resto, Aishah Alsibaee, Ainhoa Alzualde, Katherine T Andrews, Simon V Avery, Vicky M Avery, Lawrence Ayong, Mark Baker, Stephen Baker, Choukri Ben Mamoun, Sangeeta Bhatia, Quentin Bickle, Lotfi Bounaadja, Tana Bowling, Jürgen Bosch, Lauren E Boucher, Fabrice F Boyom, Jose Brea, Marian Brennan, Audrey Burton, Conor R Caffrey, Grazia Camarda, Manuela Carrasquilla, Dee Carter, Maria Belen Cassera, Ken Chih-Chien Cheng, Worathad Chindaudomsate, Anthony Chubb, Beatrice L Colon, Daisy D Colón-López, Yolanda Corbett, Gregory J Crowther, Noemi Cowan, Sarah D’Alessandro, Na Le Dang, Michael Delves, Joseph L DeRisi, Alan Y Du, Sandra Duffy, Shimaa Abd El-Salam El-Sayed, Michael T Ferdig, José A Fernández Robledo, David A Fidock, Isabelle Florent, Patrick V T Fokou, Ani Galstian, Francisco Javier Gamo, Suzanne Gokool, Ben Gold, Todd Golub, Gregory M Goldgof, Rajarshi Guha, W Armand Guiguemde, Nil Gural, R Kiplin Guy, Michael A E Hansen, Kirsten K Hanson, Andrew Hemphill, Rob Hooft van Huijsduijnen, Takaaki Horii, Paul Horrocks, Tyler B Hughes, Christopher Huston, Ikuo Igarashi, Katrin Ingram-Sieber, Maurice A Itoe, Ajit Jadhav, Amornrat Naranuntarat Jensen, Laran T Jensen, Rays H Y Jiang, Annette Kaiser, Jennifer Keiser, Thomas Ketas, Sebastien Kicka, Sunyoung Kim, Kiaran Kirk, Vidya P Kumar, Dennis E Kyle, Maria Jose Lafuente, Scott Landfear, Nathan Lee, Sukjun Lee, Adele M Lehane, Fengwu Li, David Little, Liqiong Liu, Manuel Llinás, Maria I Loza, Aristea Lubar, Leonardo Lucantoni, Isabelle Lucet, Louis Maes, Dalu Mancama, Nuha R Mansour, Sandra March, Sheena McGowan, Iset Medina Vera, Stephan Meister, Luke Mercer, Jordi Mestres, Alvine N Mfopa, Raj N Misra, Seunghyun Moon, John P Moore, Francielly Morais Rodrigues da Costa, Joachim Müller, Arantza Muriana, Stephen Nakazawa Hewitt, Bakela Nare, Carl Nathan, Nathalie Narraidoo, Sujeevi Nawaratna, Kayode K Ojo, Diana Ortiz, Gordana Panic, George Papadatos, Silvia Parapini, Kailash Patra, Ngoc Pham, Sarah Prats, David M Plouffe, Sally-Ann Poulsen, Anupam Pradhan, Celia Quevedo, Ronald J Quinn, Christopher A Rice, Mohamed Abdo Rizk, Andrea Ruecker, Robert St Onge, Rafaela Salgado Ferreira, Jasmeet Samra, Natalie G Robinett, Ulrich Schlecht, Marjorie Schmitt, Filipe Silva Villela, Francesco Silvestrini, Robert Sinden, Dennis A Smith, Thierry Soldati, Andreas Spitzmüller, Serge Maximilian Stamm, David J Sullivan, William Sullivan, Sundari Suresh, Brian M Suzuki, Yo Suzuki, S Joshua Swamidass, Donatella Taramelli, Lauve R Y Tchokouaha, Anjo Theron, David Thomas, Kathryn F Tonissen, Simon Townson, Abhai K Tripathi, Valentin Trofimov, Kenneth O Udenze, Imran Ullah, Cindy Vallieres, Edgar Vigil, Joseph M Vinetz, Phat Voong Vinh, Hoan Vu, Nao-aki Watanabe, Kate Weatherby, Pamela M White, Andrew F Wilks, Elizabeth A Winzeler, Edward Wojcik, Melanie Wree, Wesley Wu, Naoaki Yokoyama, Paul H A Zollo, Nada Abla, Benjamin Blasco, Jeremy Burrows, Benoît Laleu, Didier Leroy, Thomas Spangenberg, Timothy Wells, Paul A Willis (2016) Open source drug discovery with the Malaria Box compound collection for neglected diseases and beyond. PLOS Pathogens 12: 7. e1005763 Juli. |
B Baragaña, I Hallyburton, M C Lee, N R Norcross, R Grimaldi, T D Otto, W R Proto, A M Blagborough, S Meister, G Wirjanata, A Ruecker, L M Upton, T S Abraham, M J Almeida, A Pradhan, A Porzelle, M S Martínez, J M Bolscher, A Woodland, T Luksch, S Norval, F Zuccotto, J Thomas, F Simeons, L Stojanovski, M Osuna-Cabello, P M Brock, T S Churcher, K A Sala, S E Zakutansky, M B Jiménez-Díaz, L M Sanz, J Riley, R Basak, M Campbell, V M Avery, R W Sauerwein, K J Dechering, R Noviyanti, B Campo, J A Frearson, I Angulo-Barturen, S Ferrer-Bazaga, F J Gamo, P G Wyatt, D Leroy, P Siegl, M J Delves, D E Kyle, S Wittlin, J Marfurt, R N Price, R E Sinden, E A Winzeler, S A Charman, L Bebrevska, D W Gray, S Campbell, A H Fairlamb, P A Willis, J C Rayner, D A Fidock, K D Read, I H Gilbert (2016) Corrigendum: A novel multiple-stage antimalarial agent that inhibits protein synthesis. Nature 537: 7618. 122 May. |
|
V C Corey, A K Lukens, E S Istvan, M C S Lee, V Franco, P Magistrado, O Coburn-Flynn, T Sakata-Kato, O Fuchs, N Gnadig, G Goldgof, M Linares, M G Gomez-Lorenzo, de Cózar C, M J Lafuente-Monasterio, S Prats, S Meister, O Tanaseichuk, M Wree, Y Zhou, P Willis, F J Gamo, D E Goldberg, D A Fidock, D F Wirth, E A Winzeler (2016) A broad analysis of resistance development in the malaria parasite. Nature Communications 15: 7. 11901 June. |
N R Norcross, B Baragaña, C Wilson, I Hallyburton, M Osuna-Cabello, S Norval, J Riley, L Stojanovski, F R C Simeons, A Porzelle, R Grimaldi, S Wittlin, S Duffy, V M Avery, S Meister, L Sanz, B Jiménez-Díaz, I Angulo-Barturen, S Ferrer, M S Marínez, F J Gamo, J A Frearson, D W Gray, A H Fairlamb, E A Winzeler, D Waterson, S F Campbell, P Willis, K D Read, I H Gilbert (2016) Trisubstituted Pyrimidines as Efficacious and Fast-acting Antimalarials. Journal of Medicinal Chemistry June. |
|
J Swann, V Corey, C Scherer, N Kato, E Comer, M Maetani, Y Antonova-Koch, C Reimer, K Gagaring, M Ibanez, D Plouffe, A Zeeman, C H M Kocken, C W McNamara, S L Schreiber, B Campo, E A Winzeler, S Meister (2016) High-Throughput Luciferase-Based Assay for the Discovery of Therapeutics That Prevent Malaria. ACS Infectious Diseases 2: 4. 281–293 April. |
D M Plouffe, M Wree, A Y Du, S Meister, F Li, K Patra, A Lubar, S L Okitsu, E L Flannery, N Kato, O Tanaseichuk, E Comer, B Zhou, K Kuhen, Y Zhou, D Leroy, S L Schreiber, C A Scherer, J Vinetz, E A Winzeler (2016) High-Throughput Assay and Discovery of Small Molecules that Interrupt Malaria Transmission Cell Host & Microbe 19: 1. 114-26 Jan. |